Pyrazolo[1,5-a]-1,3,5-triazine C-nucleoside as deoxyadenosine analogue: synthesis, pairing, and resistance to hydrolysis.

نویسندگان

  • Myriam Lefoix
  • Gérald Mathis
  • Tirtsa Kleinmann
  • Jean-Christophe Truffert
  • Ulysse Asseline
چکیده

The synthesis of a pyrazolo[1,5-a]-1,3,5-triazine C-nucleoside (dA(PT)), designed to form two hydrogen bonds with a complementary dT residue, is reported. Oligonucleotides including this dA nucleoside analogue possess base-pairing properties similar to those of the parent oligonucleotide. This dA nucleoside analogue is more resistant to acid-catalyzed hydrolysis than dA.

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عنوان ژورنال:
  • The Journal of organic chemistry

دوره 79 7  شماره 

صفحات  -

تاریخ انتشار 2014